Aripiprazole Lauroxil has 13 known drug interactions based on U.S. FDA drug labeling data. 11 are classified as major interactions requiring close medical supervision. Notable interactions include combinations with Carbamazepine, Carvedilol, Clarithromycin. Patients taking Aripiprazole Lauroxil should inform their healthcare provider of all current medications — including over-the-counter drugs and supplements — to avoid potentially harmful combinations. Data sourced from OpenFDA and the NIH National Library of Medicine.
- Total
- 13
- Major
- 11
Major (11)
- Aripiprazole Lauroxil + Carbamazepine— Strong CYP3A4 inducer that decreases aripiprazole exposure. Avoid concomitant use because dosage cannot be modified.
- Aripiprazole Lauroxil + Carvedilol— Antihypertensive drug whose effect may be enhanced by aripiprazole's alpha adrenergic antagonism. Avoid concomitant use.
- Aripiprazole Lauroxil + Clarithromycin— Strong CYP3A4 inhibitor that increases aripiprazole exposure. Avoid concomitant use because dosage cannot be modified.
- Aripiprazole Lauroxil + Fluoxetine— Strong CYP2D6 inhibitor that increases aripiprazole exposure. Avoid concomitant use because dosage cannot be modified.
- Aripiprazole Lauroxil + Itraconazole— Strong CYP3A4 inhibitor that increases aripiprazole exposure. Avoid concomitant use because dosage cannot be modified.
- Aripiprazole Lauroxil + Lisinopril— Antihypertensive drug whose effect may be enhanced by aripiprazole's alpha adrenergic antagonism. Avoid concomitant use.
- Aripiprazole Lauroxil + Lorazepam— Benzodiazepine that increases sedation intensity and orthostatic hypotension when combined with aripiprazole. Avoid conc…
- Aripiprazole Lauroxil + Paroxetine— Strong CYP2D6 inhibitor that increases aripiprazole exposure. Avoid concomitant use because dosage cannot be modified.
- Aripiprazole Lauroxil + Prazosin— Antihypertensive drug whose effect may be enhanced by aripiprazole's alpha adrenergic antagonism. Avoid concomitant use.
- Aripiprazole Lauroxil + Quinidine— Strong CYP2D6 inhibitor that increases aripiprazole exposure. Avoid concomitant use because dosage cannot be modified.
- Aripiprazole Lauroxil + Rifampin— Strong CYP3A4 inducer that decreases aripiprazole exposure. Avoid concomitant use because dosage cannot be modified.