Efavirenz%2C Emtricitabine And Tenofovir Disoproxil Fumarate + Lopinavir Interaction
Contraindicatedinteraction on record
Description
( 4 , 5.4 , 7 ) • HIV-1 protease inhibitors: Coadministration of efavirenz, emtricitabine and tenofovir disoproxil fumarate with either lopinavir/ritonavir or darunavir and ritonavir increases tenofovir concentrations. Protease inhibitor: darunavir/ritonavir lopinavir/ritonavir ↑ tenofovir ↓ lopinavir ↑ tenofovir Monitor patients receiving efavirenz, emtricitabine and tenofovir disoproxil fumarate concomitantly with ritonavir-boosted darunavir for TDF-associated adverse reactions. Do not use once daily administration of lopinavir/ritonavir.
Source: FDA drug label - efavirenz, emtricitabine and tenofovir disoproxil fumarate