Itraconazole Oral Solution Containing Hydroxypropyl %CE%B2 Cyclod + Asciminib Interaction
Contraindicatedinteraction on record
Description
Concomitant use decreases asciminib Cmax and AUC, which may reduce SCEMBLIX efficacy. Avoid coadministration at all recommended doses.
Mechanism
CYP3A4 inhibition leading to decreased asciminib exposure
Source: NLP:asciminib