Fosamprenavir Calcium has 48 known drug interactions based on U.S. FDA drug labeling data. Of these, 7 are contraindicated combinations that should be avoided entirely. 3 are classified as major interactions requiring close medical supervision. Notable interactions include combinations with Alfuzosin, Esomeprazole, Lovastatin. Patients taking Fosamprenavir Calcium should inform their healthcare provider of all current medications — including over-the-counter drugs and supplements — to avoid potentially harmful combinations. Data sourced from OpenFDA and the NIH National Library of Medicine.
- Total
- 48
- Contraindicated
- 7
- Major
- 3
- Moderate
- 8
Contraindicated (7)
- Fosamprenavir Calcium + Alfuzosin— Other Agents Alpha 1-adrenoreceptor antagonist: Alfuzosin ↑Alfuzosin Coadministration is contraindicated due to potentia…
- Fosamprenavir Calcium + Esomeprazole— Proton pump inhibitors: Esomeprazole a , lansoprazole, omeprazole, pantoprazole, rabeprazole Fosamprenavir calcium: ↔ Am…
- Fosamprenavir Calcium + Lovastatin— Lipid Modifying Agents: HMG-CoA reductase inhibitors : Atorvastatin a Lovastatin, simvastatin Other lipid modifying agen…
- Fosamprenavir Calcium + Midazolam— Fosamprenavir calcium/ritonavir: ↔ Amprenavir ↔ Esomeprazole Sedative/hypnotics: Midazolam, triazolam ↑Midazolam ↑Triazo…
- Fosamprenavir Calcium + Omeprazole— Proton pump inhibitors: Esomeprazole a , lansoprazole, omeprazole, pantoprazole, rabeprazole Fosamprenavir calcium: ↔ Am…
- Fosamprenavir Calcium + Simvastatin— Lipid Modifying Agents: HMG-CoA reductase inhibitors : Atorvastatin a Lovastatin, simvastatin Other lipid modifying agen…
- Fosamprenavir Calcium + Triazolam— Fosamprenavir calcium/ritonavir: ↔ Amprenavir ↔ Esomeprazole Sedative/hypnotics: Midazolam, triazolam ↑Midazolam ↑Triazo…
Major (3)
- Fosamprenavir Calcium + Boceprevir— HCV protease inhibitor; coadministration with fosamprenavir or fosamprenavir/ritonavir is not recommended due to predict…
- Fosamprenavir Calcium + Rifampin— CYP3A4 inducer that decreases amprenavir concentrations, potentially reducing therapeutic effect of fosamprenavir.
- Fosamprenavir Calcium + Ritonavir— Potent CYP3A4 inhibitor that increases amprenavir concentrations and alters drug interaction profile; also inhibits CYP2…
Moderate (8)
- Fosamprenavir Calcium + Amlodipine— Calcium channel blockers: Diltiazem, felodipine, nifedipine, nicardipine, nimodipine, verapamil, amlodipine, nisoldipine…
- Fosamprenavir Calcium + Efavirenz— Efavirenz decreases amprenavir concentrations. Appropriate doses of unboosted combination not established; additional ri…
- Fosamprenavir Calcium + Felodipine— Calcium channel blockers: Diltiazem, felodipine, nifedipine, nicardipine, nimodipine, verapamil, amlodipine, nisoldipine…
- Fosamprenavir Calcium + Isradipine— Calcium channel blockers: Diltiazem, felodipine, nifedipine, nicardipine, nimodipine, verapamil, amlodipine, nisoldipine…
- Fosamprenavir Calcium + Nicardipine— Calcium channel blockers: Diltiazem, felodipine, nifedipine, nicardipine, nimodipine, verapamil, amlodipine, nisoldipine…
- Fosamprenavir Calcium + Nifedipine— Calcium channel blockers: Diltiazem, felodipine, nifedipine, nicardipine, nimodipine, verapamil, amlodipine, nisoldipine…
- Fosamprenavir Calcium + Nimodipine— Calcium channel blockers: Diltiazem, felodipine, nifedipine, nicardipine, nimodipine, verapamil, amlodipine, nisoldipine…
- Fosamprenavir Calcium + Nisoldipine— Calcium channel blockers: Diltiazem, felodipine, nifedipine, nicardipine, nimodipine, verapamil, amlodipine, nisoldipine…