Cyp3a Inducers + Buprenorphine Hydrochloride Interaction

Moderateinteraction on record

Description

Concomitant use decreases buprenorphine plasma concentration, potentially resulting in decreased efficacy or withdrawal syndrome. Discontinuation may cause serious respiratory depression.

Mechanism

CYP3A4 induction leading to increased metabolism

Source: NLP:buprenorphine hcl