Protease Inhibitors + Brincidofovir Interaction
Moderateinteraction on record
Description
OATP1B1/1B3 inhibitors increase brincidofovir AUC and Cmax, may increase adverse reactions. Monitor for elevations in transaminases, bilirubin, diarrhea, or GI events.
Mechanism
OATP1B1 and 1B3 inhibition
Source: NLP:brincidofovir