Protease Inhibitors + Ezetimibe And Simvastatin Interaction

Contraindicatedinteraction on record

Description

Strong CYP3A4 inhibitors that increase simvastatin plasma levels, elevating risk of myopathy and rhabdomyolysis.

Mechanism

Reduces elimination of simvastatin component via CYP3A4 inhibition

Source: NLP:ezetimibe and simvastatin