Cyp3a Inducers + Crinecerfont Interaction
Moderateinteraction on record
Description
Concomitant use decreases crinecerfont exposure, which may reduce efficacy. Requires 2-fold increase in morning and evening dosage.
Mechanism
CRENESSITY is a CYP3A4 substrate; inducers decrease its exposure
Source: NLP:crinecerfont