Cyp3a Inducers + Letrozole And Ribociclib Interaction

Majorinteraction on record

Description

Strong CYP3A4 inducers decrease ribociclib plasma exposure, potentially reducing efficacy. Coadministration should be avoided.

Mechanism

CYP3A4 induction decreases ribociclib plasma exposure

Source: NLP:letrozole and ribociclib