Desipramine + Terbinafine Interaction
Moderateinteraction on record
Description
Terbinafine inhibits CYP450 2D6, resulting in 2-fold increase in Cmax and 5-fold increase in AUC of desipramine. Effects persist up to 4 weeks after discontinuation. Monitor and may require dose reduction.
Mechanism
CYP450 2D6 inhibition
Source: NLP:terbinafine