Dextromethorphan + Terbinafine Interaction

Moderateinteraction on record

Description

Terbinafine increases dextromethorphan/dextrorphan metabolite ratio by 16- to 97-fold, converting extensive CYP2D6 metabolizers to poor metabolizer status.

Mechanism

CYP450 2D6 inhibition

Source: NLP:terbinafine