Mexiletine + Tizanidne Hydrochloride Interaction
Majorinteraction on record
Description
Should be avoided due to CYP1A2 inhibition. If necessary, initiate tizanidine at 2 mg and titrate cautiously; monitor for hypotension, bradycardia, or excessive drowsiness.
Mechanism
CYP1A2 inhibition
Source: NLP:tizanidne hydrochloride