Nefazodone + Ezetimibe And Simvastatin Interaction

Contraindicatedinteraction on record

Description

Strong CYP3A4 inhibitor that increases simvastatin plasma levels, elevating risk of myopathy and rhabdomyolysis.

Mechanism

Reduces elimination of simvastatin component via CYP3A4 inhibition

Source: NLP:ezetimibe and simvastatin