Oral Contraceptives + Tizanidine Hydrochloride Interaction
Moderateinteraction on record
Description
Moderate CYP1A2 inhibitor; concomitant use not recommended but if necessary, monitor for hypotension, bradycardia, or excessive drowsiness and reduce tizanidine dosage.
Mechanism
CYP1A2 inhibition
Source: NLP:tizanidine hydrochloride