Pioglitazone Hydrochloride + Gemfibrozil Interaction
Majorinteraction on record
Description
Strong CYP2C8 inhibitor that significantly increases pioglitazone exposure and half-life. Maximum pioglitazone dose must be limited to 15 mg daily.
Mechanism
CYP2C8 inhibition
Source: NLP:pioglitazone hydrochloride