Pioglitazone Hydrochloride + Gemfibrozil Interaction

Majorinteraction on record

Description

Strong CYP2C8 inhibitor that significantly increases pioglitazone exposure and half-life. Maximum pioglitazone dose must be limited to 15 mg daily.

Mechanism

CYP2C8 inhibition

Source: NLP:pioglitazone hydrochloride