Strong Cyp3a4 And P Glycoprotein Inducers + Lenacapavir Sodium Interaction

Majorinteraction on record

Description

Combined P-gp, UGT1A1, and strong CYP3A inhibitors may significantly increase lenacapavir plasma concentrations.

Mechanism

Inhibition of P-gp, UGT1A1, and CYP3A increases lenacapavir concentration

Source: NLP:lenacapavir sodium