Strong Inhibitors Of Cyp2d6 + Triazolam Interaction

Contraindicatedinteraction on record

Description

Concomitant use has profound effect on triazolam clearance, resulting in increased concentrations and increased risk of adverse reactions. Do not administer triazolam with strong CYP3A4 inhibitors.

Mechanism

Decreased clearance of triazolam via CYP3A4 inhibition

Source: NLP:triazolam