Talquetamab + Cyp Substrates Interaction

Majorinteraction on record

Description

Talquetamab causes cytokine release that may suppress CYP enzyme activity, resulting in increased exposure of CYP substrates. Risk is highest during step-up dosing (up to 14 days after first dose) and during/after cytokine release syndrome.

Mechanism

Cytokine-mediated suppression of CYP enzyme activity

Source: NLP:talquetamab