Amiodarone + Carvedilol Interaction
Majorinteraction on record
Description
CYP2C9 and P-glycoprotein inhibitor increases S(-)-enantiomer concentrations at least 2-fold, enhancing beta-blocking activity and potentially slowing heart rate.
Mechanism
CYP2C9 and P-glycoprotein inhibition
Source: NLP:carvedilol