Amiodarone + Macitentan And Tadalafil Interaction

Majorinteraction on record

Description

Moderate dual CYP3A4 and CYP2C9 inhibitor predicted to increase macitentan exposure. Avoid concomitant use.

Mechanism

Dual CYP3A4 and CYP2C9 inhibition

Source: NLP:macitentan and tadalafil