Amiodarone + Macitentan And Tadalafil Interaction
Majorinteraction on record
Description
Moderate dual CYP3A4 and CYP2C9 inhibitor predicted to increase macitentan exposure. Avoid concomitant use.
Mechanism
Dual CYP3A4 and CYP2C9 inhibition
Source: NLP:macitentan and tadalafil