Amiodarone + Macitentan Interaction
Contraindicatedinteraction on record
Description
Moderate dual CYP3A4 and CYP2C9 inhibitor may increase macitentan exposure. Avoid co-administration.
Mechanism
CYP3A4 and CYP2C9 inhibition
Source: NLP:macitentan
Moderate dual CYP3A4 and CYP2C9 inhibitor may increase macitentan exposure. Avoid co-administration.
CYP3A4 and CYP2C9 inhibition
Source: NLP:macitentan