Cyp3a Inducers + Imlunestrant Interaction
Majorinteraction on record
Description
Concomitant use decreases imlunestrant exposure, which may reduce effectiveness. Avoid concomitant use; if unavoidable, increase imlunestrant dosage.
Mechanism
Imlunestrant is a CYP3A substrate; strong CYP3A inducers decrease its exposure
Source: NLP:imlunestrant