Desipramine + Cinacalcet Interaction

Moderateinteraction on record

Description

CYP2D6 substrate; cinacalcet is a strong CYP2D6 inhibitor. Dose adjustment may be required for concomitant CYP2D6-metabolized medications.

Mechanism

Cinacalcet inhibits CYP2D6, increasing desipramine levels

Source: NLP:cinacalcet