Fluvoxamine + Alosetron Hydrochloride Interaction
Contraindicatedinteraction on record
Description
Fluvoxamine, a strong CYP1A2 inhibitor, increased alosetron AUC approximately 6-fold and prolonged half-life approximately 3-fold. Concomitant use is contraindicated.
Mechanism
CYP1A2 inhibition
Source: NLP:alosetron hydrochloride