Grapefruit Products + Suzetrigine Interaction
Majorinteraction on record
Description
Food or drink containing grapefruit should be avoided during treatment with JOURNAVX. Grapefruit inhibits CYP3A, increasing suzetrigine exposure.
Mechanism
Grapefruit is a CYP3A inhibitor that increases suzetrigine and M6-SUZ exposures
Source: NLP:suzetrigine