Suzetrigine + Grapefruit Products Interaction

Majorinteraction on record

Description

Food or drink containing grapefruit should be avoided during treatment with JOURNAVX. Grapefruit inhibits CYP3A, increasing suzetrigine exposure.

Mechanism

Grapefruit is a CYP3A inhibitor that increases suzetrigine and M6-SUZ exposures

Source: NLP:suzetrigine