Mao Inhibitors + Fezolinetant Interaction

Contraindicatedinteraction on record

Description

Concomitant use of CYP1A2 inhibitors increases plasma Cmax and AUC of VEOZAH. VEOZAH is contraindicated in individuals using CYP1A2 inhibitors.

Mechanism

CYP1A2 inhibition reduces VEOZAH metabolism

Source: NLP:fezolinetant