Mao Inhibitors + Ruxolitinib Interaction

Majorinteraction on record

Description

Strong inhibitors of CYP3A4 may increase ruxolitinib systemic concentrations and increase risk of adverse reactions. Concomitant use should be avoided.

Mechanism

Inhibition of CYP3A4-mediated metabolism of ruxolitinib

Source: NLP:ruxolitinib