Oral Contraceptives + Tizanidne Hydrochloride Interaction

Moderateinteraction on record

Description

Concomitant use not recommended; if necessary, monitor for hypotension, bradycardia, or excessive drowsiness and reduce or discontinue tizanidine.

Mechanism

Inhibition of CYP1A2 metabolism of tizanidine

Source: NLP:tizanidne hydrochloride