Revefenacin + Cyclosporine Interaction
Majorinteraction on record
Description
OATP1B1 and OATP1B3 inhibitor that may increase systemic exposure of revefenacin's active metabolite. Coadministration not recommended.
Mechanism
Inhibition of OATP1B1 and OATP1B3 transporters
Source: NLP:revefenacin