Sensitive Cyp3a Substrates + Suzetrigine Interaction

Moderateinteraction on record

Description

Dosage modification of sensitive CYP3A substrates may be required when initiating or discontinuing JOURNAVX. JOURNAVX is a CYP3A inducer that may reduce exposure of CYP3A substrates.

Mechanism

Suzetrigine is a CYP3A inducer that reduces exposure of sensitive CYP3A substrates

Source: NLP:suzetrigine