Leucovorin + Irinotecan Hydrochloride Interaction

Moderateinteraction on record

Description

Co-administration with 5-FU reduces SN-38 Cmax by 14% and AUC by 8%. This sequence is recommended in combination trials.

Mechanism

Reduced active metabolite exposure when irinotecan followed by 5-FU and leucovorin

Source: NLP:irinotecan hydrochloride