Mao Inhibitors + Elagolix And Estradiol And Norethisterone Interaction
Contraindicatedinteraction on record
Description
OATP1B1 inhibitors that significantly increase elagolix plasma concentrations are contraindicated due to increased risk of elagolix-associated adverse reactions.
Mechanism
OATP1B1 inhibition
Source: NLP:elagolix and estradiol and norethisterone