P Gp Or Bcrp Substrates + Berotralstat Hydrochloride Interaction
Majorinteraction on record
Description
P-gp inducers may decrease berotralstat plasma concentration, leading to reduced efficacy of ORLADEYO. Avoid concomitant use.
Mechanism
Berotralstat is a substrate of P-gp; inducers decrease plasma concentration
Source: NLP:berotralstat hydrochloride